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 2-methyl-1-(phenylsulfonyl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-Pyrrolo[2,3-b]pyridine (5-(((tert-Butoxycarbonyl)amino)-methyl)furan-2-yl)boronic acid 1-(3-aminophenyl)-4-Piperidinol tert-butyl 3-bromo-5-fluoropyridine-4-carboxylate
 B-(3-chlorobiphenyl]-3-yl)Boronic acid 1-cyclopentyl-1H-Pyrazol-4-amine 1-(2-fluorophenyl)-1H-Pyrazol-4-amine 4-methylpyridine-2-carboxamidine hydrochloride
 5-(tetrahydro-3-furanyl)-1H-Pyrazol-3-amine tert-butyl dibut-3-enylcarbamate 5-methyl-4-Oxazolecarbonitrile 4-methyl-2-Oxazolecarbonitrile
 5-methyl-4-Oxazolecarboxamide 4-methyl-2-Thiazolecarboximidamide 4-chloro-2-(2-thienyl)-1H-Pyrrolo[2,3-b]pyridine 4-cyclopropyl-2-Thiazolecarbonitrile
 B-7-benzofuranylBoronic acid tert-butyl 3-(phenylcarbamoyl)pyrrolidin-3-ylcarbamate tert-butyl 4-cyclopropylthiazol-2-ylcarbamate 5-methyl-4-Oxazolecarboximidamide
 3-methyl-3-Morpholinecarboxylic acid Pyrazolo[1,5-a]pyridin-6-amine 5-chloro-Imidazo[2,1-b]thiazole-6-carboxylic acid 4-cyclopropylthiazole-2-carboxamidine hydrochloride
 4-tert-butylthiazole-2-carboxamidine hydrochloride 1,4-dimethyl-1H-imidazole-2-carboxamidine hydrochloride tert-butyl 3-carbamoylpyrrolidin-3-ylcarbamate benzyl 4-hydroxy-3-(hydroxymethyl)piperidine-1-carboxylate
 2-methyl-1H-Pyrrolo[2,3-b]pyridine-4-carbonitrile 1H-Pyrrolo[2,3-b]pyridine-4-carboximidamide tert-butyl 4-(3-amino-1-isopropyl-1H-pyrazol-5-yl)piperidine-1-carboxylate N,3-dimethoxy-N,2,2-trimethylPropanamide
 tert-butyl 4-(3-amino-1-cyclopentyl-1H-pyrazol-5-yl)piperidine-1-carboxylate 4-cyclopropyl-5-(4-piperidinyl)-2-Thiazolamine 6-cyclopropyl-2-fluoro-3-Pyridinamine 2-fluoro-6-(4-morpholinyl)-3-Pyridinamine
 2-cyclopropyl-1H-Pyrrolo[2,3-b]pyridine-4-carboximidamide tert-butyl 4-(5-(1,3-dioxoisoindolin-2-yl)-1H-pyrazol-3-yl)piperidine-1-carboxylate tert-butyl 4-(1-isopropyl-3-(1,3-dioxoisoindolin-2-yl)-1H-pyrazol-5-yl)piperidine-1-carboxylate tert-butyl 4-(5-iodo-1H-pyrazol-3-yl)piperidine-1-carboxylate
 tert-butyl 4-(3-iodo-1-(3-oxocyclopentyl)-1H-pyrazol-5-yl)piperidine-1-carboxylate tert-butyl 4-(1-(tetrahydrofuran-3-yl)-3-iodo-1H-pyrazol-5-yl)piperidine-1-carboxylate 3-iodo-5-(tetrahydro-3-furanyl)-1H-Pyrazole 5-bromo-2-(4-pyridinyl)-Pyrido[3,4-d]pyrimidin-4(3H)-one
 tert-butyl 4-(1-(cyclobutylmethyl)-3-(1,3-dioxoisoindolin-2-yl)-1H-pyrazol-5-yl)piperidine-1-carboxylate tert-butyl 3-(1-cyclopentyl-3-(1,3-dioxoisoindolin-2-yl)-1H-pyrazol-5-yl)azetidine-1-carboxylate tert-butyl 4-(3-amino-1-(cyclobutylmethyl)-1H-pyrazol-5-yl)piperidine-1-carboxylate tert-butyl 3-(3-amino-1-cyclopentyl-1H-pyrazol-5-yl)azetidine-1-carboxylate
 tert-butyl 4-(5-(2,5-dimethyl-1H-pyrrol-1-yl)-1H-pyrazol-3-yl)piperidine-1-carboxylate tert-butyl 4-(1-cyclopentyl-3-(2,5-dimethyl-1H-pyrrol-1-yl)-1H-pyrazol-5-yl)piperidine-1-carboxylate tert-butyl 3-(5-iodo-1H-pyrazol-3-yl)pyrrolidine-1-carboxylate tert-butyl 4-(1-(tetrahydro-2H-pyran-4-yl)-3-iodo-1H-pyrazol-5-yl)piperidine-1-carboxylate
 tert-butyl 3-(1-cyclopentyl-3-iodo-1H-pyrazol-5-yl)pyrrolidine-1-carboxylate 1-cyclopentyl-3-iodo-5-(tetrahydro-3-furanyl)-1H-Pyrazole tert-butyl 5-chloro-4-cyclopropylthiazol-2-ylcarbamate 4-cyclopropyl-5-[1-(3-oxetanyl)-4-piperidinyl]-2-Thiazolamine
 2-cyclopentyl-4,5-diiodo-1H-Imidazole 2-cyclopentyl-5-iodo-1H-Imidazole tert-butyl 4-(2-cyclopentyl-4-iodo-1H-imidazol-1-yl)piperidine-1-carboxylate 2-(4-pyridinyl)-Pyrido[3,4-d]pyrimidin-4(3H)-one
 4-chloro-2-(4-pyridinyl)-Pyrido[3,4-d]pyrimidine 5-methoxy-2-(4-pyridinyl)-Pyrido[3,4-d]pyrimidin-4(3H)-one 4-isopropylthiazole-2-carboxamidine hydrochloride 4-bromo-2-(diethoxymethyl)Thiazole
 4-(4-morpholinyl)-2-(4-pyridinyl)-Pyrido[3,4-d]pyrimidine 8-chloro-4-(1-piperazinyl)-2-(4-pyridinyl)-Pyrido[3,4-d]pyrimidine di-tert-butyl 2-ethynylpiperazine-1,4-dicarboxylate ethyl 5-chloroimidazo[2,1-b]thiazole-6-carboxylate
 ethyl 3-isobutylimidazo[2,1-b]thiazole-6-carboxylate 2-(2-thienyl)-1H-Pyrrolo[2,3-b]pyridine-4-carbonitrile 2-Bromo-4-isopropoxy-5-nitrotoluene 2-Bromo-4-isopropoxy-1-methylbenzene
 ethyl 5-(1-hydroxy-2-(piperidin-1-yl)ethyl)-1H-indole-2-carboxylate 4-methyl-2-(2-pyrimidinyl)Benzoic acid B-[1-(2-hydroxy-2-methylpropyl)-3-methyl-1H-pyrazol-4-yl]Boronic acid 5-methyl-2-(1-methyl-1H-pyrazol-3-yl)Benzoic acid
 5-methyl-2-(5-thiazolyl)Benzoic acid 5-methyl-2-(2-methyl-4-pyridinyl)Benzoic acid 2-(2-methoxy-5-pyrimidinyl)-5-methylBenzoic acid 5-methyl-2-(3-pyridazinyl)Benzoic acid
 5-oxo-1-Oxa-4,9-diazaspiro[5.5]undecane-9-carboxylic acid 1,1-dimethylethyl ester 6-(2,8-diazaspiro[4.5]dec-2-yl)-3-Pyridinecarbonitrile 2-[4-(methylsulfonyl)phenyl]-2,8-Diazaspiro[4.5]decane 3-bromo-6-(methylsulfonyl)Pyridazine
 5-(2,8-diazaspiro[4.5]dec-2-yl)-3-Pyridinecarbonitrile 2-(2,8-diazaspiro[4.5]dec-2-yl)-4-Pyridinecarbonitrile 4-(2,8-diazaspiro[4.5]dec-2-yl)-2-Pyridinecarbonitrile tert-butyl 3-(hydroxymethyl)-3-methoxypyrrolidine-1-carboxylate
 tert-butyl 4-(2-chlorobenzyl)-4-formylpiperidine-1-carboxylate tert-butyl 4-(4-(trifluoromethyl)phenyl)-4-(hydroxymethyl)piperidine-1-carboxylate tert-butyl 4-(4-(trifluoromethyl)phenyl)-4-formylpiperidine-1-carboxylate 4-ethoxy-3-nitroBenzoic acid
 (2S)-2-amino-3-mercaptobutanoic acid (2R)-2-amino-2-methyl-3-sulfanylpropanoic acid hydrochloride (2S)-2-amino-2-methyl-3-sulfanylpropanoic acid hydrochloride methyl 5-(((S)-2-((tert-butoxycarbonyl)amino)-3- (4-carbamoyl-2,6-dimethylphenyl)-N-((S)-1-(4- phenyl-1H-imidazol-2- yl)ethyl)propanamido)methyl)-2-methoxybenzoate
 3-(4-phenoxyphenyl)-1-(3R)-3-piperidinyl-1H-Pyrazolo[3,4-d]pyrimidin-4-amine dihydrochloride 4-ethoxy-3-(trifluoromethyl)Benzoic acid 3-cyano-5-(trifluoromethoxy)Benzoic acid 1-(5-amino-5,6,7,8-tetrahydro-2-naphthalenyl)Ethanone
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